Overview

  • Product name
    (+)-JQ1
  • Description
    Potent, selective and cell-permeable BET bromodomain inhibitor
  • Alternative names
    • (S)-(+)-tert-Butyl 2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate
    • 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-trimethyl-, 1,1-dimethylethyl ester, (6S)-
  • Biological description

    Potent, selective and cell-permeable BET bromodomain inhibitor (Kd values are 50 and 90 nM at BRD4 first and second bromodomains, respectively).

  • Purity
    > 99%

Properties

References

This product has been referenced in:

See 1 Publication for this product

Customer reviews and Q&As


Te confirmo que el producto ab141498 solo se suministra como enantiómero positivo, que es el enantiómero activo que actúa como potente inhibidor de BET. Podría consultar con el laboratorio si fuera posible aislar el isómero negativo, o la mezcla r...

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Please note: All products are "FOR RESEARCH USE ONLY AND ARE NOT INTENDED FOR DIAGNOSTIC OR THERAPEUTIC USE, NOT FOR USE IN HUMANS"

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