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We have 451 products in: Biochemicals >> Pharmacology >> Enzymes

Enzyme modulators beginning with A - B

A - B   C - D   E - I   J - M   N - P   Q - S   T - Z   0 - 9   

Code

Name

Details

 Image Abreview Publication 

Asc-335  

A 769662 

AMP-activated protein kinase activator

Purity: > 99%

 
Specific publication references
 
 
 

A771726 (Teriflunomide) 

Active metabolite of leflunomide. Dihydroorotate dehydrogenase inhibitor.

Purity: > 98%

 
 
 
 
Asc-350  

AACOCF3 (Arachidonyl trifluoromethyl ketone) 

Phospholipase-A2 inhibitor

Purity: > 98%

 
 
 
 
Asc-860  

(+)-Abscisic acid 

Phytohormone; produced by a variety of cells in humans and animals

Purity: > 99%

 
 
 
 

Ac-IEPD-CHO 

Reversible granzyme B and caspase-8 inhibitor

Purity: > 95%

 
 
 
 
  

Acarbose 

Potent α-glucosidase inhibitor

Purity: > 98%

 
 
 
 
Asc-990  

Acetaminophen 

Selective COX-3 inhibitor

Purity: > 98%

 
 
 
 
  

Acivicin 

γ-glutamyl transpeptidase inhibitor

Purity: > 98%

 
 
 
 

Aclacinomycin A 

Topoisomerase I and II inhibitor

Purity: > 95%

 
 
 
 
Asc-631  

Acyclovir 

Inhibits viral DNA polymerase. Antiherpetic agent

Purity: > 99%

 
 
 
 
Asc-493  

Adenosine 3′,5′-cyclic monophosphate (cAMP) 

Second messenger. PKA activator.

Purity: > 98%

 
 
 
 

AG-126 

Tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 

AG-1288 

Non-selective tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 

AG-370 

Selective PDGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
Asc-1170  

AG 1296 

Potent specific PDGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
Asc-950  

AG 490 

JAK2/3 inhibitor

Purity: > 99%

 
 
 
 

AGK2 

Selective reversible cell-permeable sirtuin2 (SIRT2) inhibitor

Purity: > 95%

 
 
 
 
Asc-358  

AICAR (Acadesine/AICA riboside) 

Cell-permeable activator of AMP-activated protein kinase

Purity: > 98%

Images
 
 
 
 

Akt Inhibitor, Isozyme-Selective 

Potent isozyme selective Akt1/2 kinase inhibitor

Purity: > 97%

 
 
 
 

ALLM 

Calpain and cathepsin inhibitor

Purity: > 95%

 
 
 
 

ALLN 

Calpain inhibitor

Purity: > 95%

 
 
 
 

AMI-1 

Potent, selective and reversible protein arginine methyltransferase inhibitor

Purity: > 98%

 
 
 
 
Asc-1069  

3-Aminobenzamide (3-AB) 

PARP inhibitor

Purity: > 99%

 
 
 
 
Asc-123  

Aminoguanidine hydrochloride 

NOS inhibitor

Purity: > 98%

 
 
 
 
  

4-Aminophenyl phosphate monosodium salt 

Alkaline phosphatase substrate

Purity: > 97%

 
 
 
 
Asc-495  

Anisomycin 

Protein synthesis inhibitor

Purity: > 98%

Images
 
 
 
 

Apicidin 

Potent HDAC inhibitor

Purity: > 95%

 
 
 
 
Asc-615  

Apocynin 

Selective NADPH-oxidase inhibitor

Purity: > 99%

Images
 
 
 
 
Asc-1227  

Apoptosis Activator 2 (AAII) 

Cytochrome c caspase activator and apoptosis inducer

Purity: > 99%

 
 
 
 
Asc-1295  

AR-A014418 

Highly selective GSK-3 inhibitor

Purity: > 99%

 
 
 
 

Arachidonoyl-AMC 

Fluorogenic substrate for fatty acid amide hydrolase (FAAH)

Purity: > 99%

 
 
 
 
  

AS-041164 

Potent and selective PI3Kγ inhibitor

Purity: > 98%

 
 
 
 
  

AS-252424 

Potent and selective PI3Kγ inhibitor

Purity: > 95%

 
 
 
 
  

AS-604850 

Selective, ATP-competitive PI3Kγ inhibitor

Purity: > 98%

 
 
 
 
  

AS-605240 

Potent and selective PI3Kγ inhibitor

Purity: > 98%

 
 
 
 
Asc-1016  

Ascomycin 

Calcineurin/PP2B inhibitor. Immunosuppressant and antifungal activity.

Purity: > 98%

 
 
 
 
Asc-1083  

Atorvastatin hemicalcium salt 

Potent HMG-CoA reductase inhibitor

Purity: > 99%

Images
 
 
 
 

AUDA 

Potent epoxide hydrolase inhibitor. Antihypertensive.

Purity: > 98%

 
 
 
 
Asc-1027  

Aurintricarboxylic acid (ATA) 

Apoptosis inhibitor

 
 
 
 

AZ-960 

Novel, potent and selective JAK2 inhibitor

Purity: > 95%

 
 
 
 
Asc-842  

5-Aza-2'-deoxycytidine (Decitabine) 

Potent DNA methyltransferase inhibitor; epigenetic modifier

Purity: > 99%

 
 
 
 

B2 

Potent SIRT2 inhibitor

Purity: > 95%

 
 
 
 
Asc-497  

Bafilomycin A1 

Highly potent, selective (V)-ATPase inhibitor

Purity: > 98%

 
Specific publication references
 
 
 
Asc-723  

Baicalein 

Flavonoid. Lipoxygenase inhibitor.

Purity: > 98%

Images
 
 
 
 

Batimastat (BB-94) 

Potent, broad-spectrum MMP inhibitor

Purity: > 98%

 
 
 
 

Bay 61-3606 hydrochloride 

Potent, selective, cell-permeable Syk kinase inhibitor

Purity: > 98%

 
 
 
 
Asc-1166  

Benazepril hydrochloride 

Angiotensin-converting enzyme (ACE) inhibitor. Prodrug.

Purity: > 99%

 
 
 
 

Bestatin 

Aminopeptidase inhibitor; immunomodulator

Purity: > 99%

 
 
 
 

Bikinin 

Cell-permeable, ATP-competitive 7 Arabidopsis GSK-3 inhibitor

Purity: > 95%

 
 
 
 

Biotin-DEVD-FMK 

Biotin-conjugated, potent, irreversible caspase-3 inhibitor. Cell-permeable.

Purity: > 95%

 
 
 
 

Biotin-IETD-FMK 

Biotinylated, irreversible caspase-8 inhibitor

Purity: > 95%

 
 
 
 

Biotin-VAD-FMK 

Pan-caspase inhibitor

Purity: > 95%

 
 
 
 
Asc-976  

Bisdemethoxycurcumin 

Apoptotic anti-cancer, anti-inflammatory and anti-oxidant curcuminoid

Purity: > 98%

 
 
 
 

BIX 01294 

Potent G9a and G9a-like protein histone lysine methyltransferase inhibitor

Purity: > 95%

 
 
 
 

BML-210 

HDAC inhibitor

Purity: > 98%

 
 
 
 

BML-244 

Potent cathepsin K inhibitor

Purity: > 98%

 
 
 
 

BML-259 

Potent Cdk5/p25 and Cdk2 inhibitor

Purity: > 98%

 
 
 
 

Boc-D-FMK 

Irreversible general caspase inhibitor. Cell-permeable.

Purity: > 95%

 
 
 
 

Boc-Gly-Val-Val-CHO (Boc-GVV-CH) 

Substrate based inhibitor of γ-secretase (γ-40 site)

Purity: > 98%

 
 
 
 

BPPA 

Telomerase inhibitor

Purity: > 97%

 
 
 
 

bpV(phen) 

Potent protein phosphotyrosine phosphatase inhibitor. PTEN inhibitor.

Purity: > 98%

 
 
 
 

BRL-50481 

Selective PDE7 inhibitor

Purity: > 98%

 
 
 
 
Asc-616  

2,3-Butanedione 2-monoxime (BDM) 

Non-selective myosin ATPase inhibitor

 
 
 
 

Butyrolactone I 

Cell permeable, selective, ATP-competitive cyclin-dependent kinase (CDK) inhibitor

Purity: > 99%

 
 
 
 
Asc-1255  

Butyrolactone 3 

Histone acetyltransferase Gcn5 inhibitor

Purity: > 99%

 
 
 
 
Asc-1304  

BVT 948 

Non-competitive, irreversible protein tyrosine phosphatase (PTP) inhibitor

Purity: > 99%

 
 
 
 

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A - B   C - D   E - I   J - M   N - P   Q - S   T - Z   0 - 9   

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