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Adrenoceptors

Code

Name

Details

 Image Abreview Publication 

(S)-Carazolol Fluorescent ligand (Red) 

Fluorescent β3 adrenoceptor agonist

Purity: > 97%

Images
 
 
 
 

(S)-Propranolol Fluorescent ligand (Red) 

Fluorescent β2 adrenoceptor antagonist

Purity: > 97%

Images
 
 
 
 

Alprenolol Fluorescent ligand (Red) 

Fluorescent β2 adrenoceptor antagonist

Purity: > 97%

Images
 
 
 
 
Asc-576  

Asenapine maleate 

Multiple receptor antagonist. Anti-psychotic agent.

Purity: > 99%

 
 
 
 
Asc-752  

(R,S)-Atenolol 

β1 adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-856  

(S)-(-)-Atenolol 

Selective β1 adrenoceptor antagonist

Purity: > 98%

 
Specific publication references
 
 
 
Asc-785  

Atipamezole hydrochloride 

Selective α2 adrenergic receptor antagonist

Purity: > 99%

 
 
 
 
Asc-783  

(±)-Bisoprolol hemifumarate 

Selective β1 antagonist

Purity: > 99%

 
 
 
 
Asc-520  

BMY 7378 dihydrochloride 

5-HT1A partial agonist. α-adrenoceptor antagonist.

Purity: > 99%

 
 
 
 

Bopindolol malonate 

Non-selective, potent adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-806  

BRL 44408 maleate 

Selective α2A adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-534  

Bupropion hydrochloride 

Non-selective DAT/NET inhibitor

Purity: > 98%

 
 
 
 
Asc-709  

Carvedilol 

Potent β and α1-adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-729  

(±)-Chlorpheniramine maleate 

Potent H1 antagonist and SNRI

Purity: > 99%

 
 
 
 
Asc-730  

Chlorpromazine hydrochloride 

Typical antipsychotic. Non-selective receptor antagonist.

Purity: > 99%

 
 
 
 
Asc-954  

Cimaterol 

β-adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-753  

Clonidine hydrochloride 

α2 adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-768  

Dobutamine hydrochloride 

β1 and β2 adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-754  

Doxazosin mesylate 

Selective α1-adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-786  

Formoterol hemifumarate 

Potent long-acting β2-adrenergic receptor agonist

Purity: > 99%

 
 
 
 
Asc-808  

ICI 118551 hydrochloride 

Highly selective β2 adrenergic receptor antagonist

Purity: > 99%

 
 
 
 
Asc-1130  

Idazoxan hydrochloride 

α2-adrenoceptor antagonist and I2 ligand

Purity: > 99%

 
 
 
 
Asc-1046  

Imipramine hydrochloride 

Tricyclic antidepressant

Purity: > 98%

 
 
 
 
Asc-710  

Isoprenaline hydrochloride 

Non selective β-adrenoceptor agonist

Purity: > 99%

Images
 
 
 
 

Isotetrandrine 

Cell-permeable PLA2 inhibitor

Purity: > 98%

 
 
 
 
Asc-1129  

JP1302 dihydrochloride 

Potent and selective α2C antagonist

Purity: > 99%

 
 
 
 
Asc-769  

Maprotiline hydrochloride 

Noradrenaline reuptake inhibitor

Purity: > 99%

 
 
 
 
Asc-711  

Metoprolol tartrate 

β1-adrenergic receptor antagonist

Purity: > 99%

 
 
 
 
Asc-788  

Mianserin hydrochloride 

Multiple receptor antagonist. Activity at 5-HT2, H1 and α2 receptors.

Purity: > 99%

 
 
 
 
Asc-755  

Milnacipran hydrochloride 

Serotonin and norepinephrine reuptake inhibitor

Purity: > 99%

 
 
 
 
Asc-068  

Mirtazapine 

Antidepressant. α2, 5-HT2, 5-HT3 antagonist.

Purity: > 99%

 
 
 
 
Asc-789  

Moxonidine hydrochloride 

I1 imidazoline receptor and α2 adrenergic agonist

Purity: > 99%

 
 
 
 
Asc-756  

Naftopidil hydrochloride 

α1 adrenergic receptor antagonist

Purity: > 98%

 
 
 
 
Asc-543  

NAN-190 hydrobromide 

Potent 5-HT1A antagonist

Purity: > 99%

 
 
 
 
Asc-790  

Nebivolol hydrochloride 

Selective β1 antagonist

Purity: > 99%

 
 
 
 
Asc-587  

Nefazodone hydrochloride 

Potent 5-HT2A antagonist

Purity: > 99%

 
 
 
 
Asc-1134  

Nisoxetine hydrochloride 

Potent and selective norepinephrine reuptake (NET) inhibitor

Purity: > 99%

 
 
 
 
Asc-717  

L-(-)-Norepinephrine-(+)-bitartrate (Noradrenaline) 

Endogenous α adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-770  

Octopamine hydrochloride 

Full β3 agonist: invertebrate biogenic amine

Purity: > 99%

 
 
 
 
Asc-736  

Olanzapine 

Non-selective 5-HT, dopamine, histamine and muscarinic antagonist.

Purity: > 99%

Images
 
 
 
 
Asc-712  

Oxymetazoline hydrochloride 

α1A and partial α2A adrenoceptor agonist.

Purity: > 99%

 
 
 
 

Phentolamine hydrochloride 

Non-selective α antagonist

Purity: > 98%

 
Specific publication references
 
 
 
Asc-761  

(R)-(-)-Phenylephrine hydrochloride 

α1 adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-521  

Pindolol 

5-HT1A and 5-HT1B receptor antagonist

Purity: > 99%

 
 
 
 

Pindolol Fluorescent ligand (Red) 

Fluorescent β2 antagonist

Purity: > 97%

Images
 
 
 
 
Asc-238  

Prazosin hydrochloride 

α-adrenoceptor antagonist. Melatonin antagonist.

Purity: > 99%

 
Specific publication references
 
 
 

Propranolol Fluorescent ligand (Red) 

Fluorescent β2 adrenoceptor antagonist

Purity: > 97%

Images
 
 
 
 

(S)-Propranolol Fluorescent Ligand (green) 

Fluorescent ß2 adrenoceptor antagonist

Purity: > 97%

Images
 
 
 
 
Asc-757  

Propranolol hydrochloride 

Potent β-adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-1133  

(S)-Propranolol hydrochloride 

Non-selective β-adrenoceptor antagonist

Purity: > 98%

 
 
 
 
Asc-875  

Rauwolscine hydrochloride 

Potent α2 adrenergic antagonist

Purity: > 99%

 
 
 
 
Asc-157  

Reboxetine mesylate 

Noradrenaline reuptake inhibitor

Purity: > 99%

 
 
 
 
Asc-601  

Rotigotine hydrochloride 

Dopamine receptor agonist

Purity: > 99%

 
 
 
 

Salbutamol Fluorescent ligand (Red) 

Fluorescent β2 adrenoceptor agonist

Purity: > 97%

Images
 
 
 
 
Asc-714  

Salbutamol hemisulfate 

Non-selective β-adrenoceptor agonist

Purity: > 99%

 
 
 
 
Asc-529  

Sibutramine hydrochloride 

Serotonin, noradrenaline & dopamine re-uptake inhibitor

Purity: > 98%

 
 
 
 

Sotalol hydrochloride 

Non-selective beta adrenoceptor antagonist and potassium channel blocker

Purity: > 98%

 
 
 
 
Asc-1135  

SR 59230A hydrochloride 

Potent, selective β3-adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-792  

Terbutaline hemisulfate 

Selective β2 receptor agonist

Purity: > 99%

 
 
 
 
Asc-784  

(S)-Timolol maleate 

Potent non-selective β-adrenoceptor antagonist

Purity: > 99%

 
 
 
 
Asc-758  

(R)-Tomoxetine hydrochloride 

Potent, selective norepinephrine reuptake inhibitor

Purity: > 99%

 
 
 
 
Asc-773  

UK 14,304 tartrate 

Selective α2 adrenergic agonist

Purity: > 99%

 
 
 
 
Asc-715  

Venlafaxine hydrochloride 

Serotonin-norepinephrine reuptake inhibitor

Purity: > 99%

 
 
 
 
Asc-759  

Xylazine hydrochloride 

α2 adrenergic receptor agonist

Purity: > 99%

 
 
 
 
Asc-239  

Yohimbine hydrochloride 

Selective α2-adrenoceptor antagonist

Purity: > 98%

 
Specific publication references