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Nuclear Receptors

Code

Name

Details

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Tibolone 

A synthetic normethyltestosterone derivative used in the prevention of postmenopaual osteoporosis. It is capable of inducing apoptosis in breast cancer cell lines.

Purity: > 98%

 
 
 
 

Adapalene 

Selective RARβ and RARγ agonist

Purity: > 98%

 
 
 
 
Asc-1024  

AM 80 

Selective retinoic acid receptor α/β (RARα/β) agonist

Purity: > 98%

 
 
 
 
Asc-1285  

4-Androstene-3,17-dione (Androstenedione) 

Testosterone precursor. Major endogenous androgen.

Purity: > 99%

 
 
 
 

Auraptene 

Activates PPARα and PPARγ. Modulates estrogen receptors

Purity: > 98%

 
 
 
 
Asc-1280  

Betamethasone valerate 

Potent glucocorticoid; immunomodulator

Purity: > 98%

 
 
 
 
Asc-1025  

Bexarotene 

Potent RXR agonist

Purity: > 99%

 
 
 
 
Asc-1233  

Bezafibrate 

Pan-PPAR agonist

Purity: > 99%

 
 
 
 
Asc-1249  

Bicalutamide (ICI176334) 

Non-steroidal, competitive androgen receptor antagonist

Purity: > 99%

 
 
 
 
Asc-1139  

Ciglitazone 

Selective PPARγ agonist

Purity: > 98%

 
 
 
 
Asc-1331  

Clofibrate 

PPARα agonist

Purity: > 99%

 
 
 
 
Asc-833  

Clofibric acid 

PPARα agonist

Purity: > 99%

 
 
 
 
Asc-1183  

Clomiphene citrate 

Selective estrogen receptor modulator (SERM)

Purity: > 98%

 
 
 
 
Asc-391  

Daidzein 

Phytoestrogen

Purity: > 99%

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Specific publication references
 
 
 
Asc-743  

Dexamethasone 

Anti-inflammatory glucocorticoid

Purity: > 99%

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Asc-1282  

Dienogest 

Steroidal progesterone

Purity: > 99%

 
 
 
 
Asc-166  

DPN 

Potent, selective ERβ agonist

Purity: > 99%

 
 
 
 
Asc-1251  

Eplerenone 

Selective mineralocorticoid antagonist

Purity: > 99%

 
 
 
 
Asc-390  

Equol 

Metabolite of phytoestrogen daidzein

Purity: > 99%

 
 
 
 
Asc-657  

17β-Estradiol 

Selective agonist of ER receptor

Purity: > 99%

 
 
 
 
Asc-832  

Fenofibrate 

Potent, selective PPAR-α agonist

Purity: > 99%

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Asc-1277  

Finasteride 

Selective type II 5α-reductase inhibitor

Purity: > 99%

 
 
 
 
Asc-1234  

Flutamide 

Non-steroidal, competitive androgen receptor antagonist

Purity: > 99%

 
 
 
 
Asc-1281  

Fluticasone propionate 

Potent, selective glucocorticoid agonist

Purity: > 99%

 
 
 
 

G3335 

Selective, cell-permeable, reversible PPARγ antagonist.

Purity: > 97%

 
 
 
 
Asc-826  

GSK 4716 

Selective ERRβγ agonist

Purity: > 99%

 
 
 
 

GW1929 

Potent, selective PPARγ agonist

Purity: > 98%

 
 
 
 
Asc-1125  

GW 9662 

Selective PPARγ antagonist

Purity: > 99%

 
 
 
 
Asc-1261  

GW 9662-d5 

Potent, irreversible and selective PPARγ antagonist

Purity: > 99%

 
 
 
 
Asc-1250  

Hydrocortisone 

Adrenal glucocorticoid; immunosuppressant

Purity: > 99%

 
 
 
 

(Z)-4-Hydroxytamoxifen 

Potent and selective estrogen receptor modulator

Purity: > 98%

 
 
 
 
Asc-131  

ICI 182,780 

Estrogen receptor antagonist

Purity: > 99%

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Asc-719  

Indomethacin 

Non-selective COX inhibitor

Purity: > 99%

 
 
 
 
Asc-1293  

Letrozole 

Highly potent, reversible, selective aromatase inhibitor

Purity: > 99%

 
 
 
 

Luffariellolide 

Potent phospholipase A2 (PLA2) inhibitor. Agonist at RARα

Purity: > 98%

 
 
 
 

Methoprene acid 

Specific RXR activator

Purity: > 98%

 
 
 
 
Asc-356  

Mifepristone (RU486) 

PR and GR antagonist

Purity: > 98%

 
 
 
 
Asc-1140  

MK886 

Potent lipoxygenase inhibitor

Purity: > 98%

 
 
 
 

13-OXO-ODE (13-Keto-octadeca-9Z,11E-dienoic acid) 

Potent PPARα agonist

Purity: > 98%

 
 
 
 
Asc-794  

Pioglitazone hydrochloride 

Selective PPAR-γ agonist

Purity: > 99%

 
 
 
 

Potassium canrenoate 

Aldosterone antagonist

Purity: > 98%

 
 
 
 
Asc-161  

PPT 

Subtype selective ERα agonist

Purity: > 99%

 
 
 
 

Prednisolone sodium phosphate 

Water-soluble glucocorticoid

Purity: > 98%

 
 
 
 

Prednisone 

Glucocorticoid. Immunosuppressant an anti-inflammatory agent.

Purity: > 98%

 
 
 
 

Prednisone Acetate 

Glucocorticoid. Anti-inflammatory agent.

Purity: > 98%

 
 
 
 
Asc-1252  

Progesterone 

Endogenous progesterone receptor agonist

Purity: > 99%

 
 
 
 
Asc-1023  

9-cis-Retinoic acid 

High affinity, endogenous retinoic acid receptor agonist

Purity: > 98%

 
 
 
 

all-trans Retinol (Vitamin A) 

Retinoic acid receptor ligand

Purity: > 98%

 
 
 
 

Retinyl acetate 

Retinol derivative, vitamin A analog. Anticarcinogenic and apoptotic agent

Purity: > 98%

 
 
 
 

Retinyl palmitate 

Vitamin A analog. Storage ester of retinol. Antitumor agent.

 
 
 
 

Ro 41-5253 

Potent, selective retinoic acid receptor antagonist

Purity: > 99%

 
 
 
 
Asc-762  

Rosiglitazone 

Selective PPARγ agonist

Purity: > 99%

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Asc-1289  

Spironolactone 

Mineralocorticoid receptor antagonist

Purity: > 99%

 
 
 
 

SR1001 

Specific RORα and RORγt antagonist

Purity: > 98%

 
 
 
 

SR-12813 

Potent, selective PXR agonist

Purity: > 98%

 
 
 
 

Stanozolol 

Synthetic anabolic steroid derived from dihydrotestosterone

Purity: > 98%

 
 
 
 
  

T0070907 

Potent, selective PPARγ antagonist

Purity: > 98%

 
 
 
 
Asc-656  

Tamoxifen citrate 

Estrogen receptor antagonist and partial agonist

Purity: > 99%

 
 
 
 
Asc-1294  

TCPOBOP 

Potent murine constitutive androstane receptor (mCAR) agonist

Purity: > 99%

 
 
 
 
Asc-831  

Telmisartan 

Selective angiotensin II (AT1) antagonist

Purity: > 99%

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Tetradecylthioacetic acid 

3-Thia synthetic fatty acid. Pan-PPAR activator.

Purity: > 98%

 
 
 
 

WAY-200070 

Potent, selective ERβ agonist

Purity: > 98%