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Purinergic receptors

Code

Name

Details

 Image Abreview Publication 

Asc-413  

A 438079 

Potent, competitive P2X7 receptor antagonist

Purity: > 98%

 
 
 
 
Asc-498  

Adenosine 

Endogenous P1 receptor agonist

Purity: > 99%

 
 
 
 
Asc-385  

ATP disodium salt 

P2 receptor agonist. Signalling molecule.

Purity: > 99%

 
Specific publication references
 
 
 
Asc-389  

Brilliant Blue G 

Potent, noncompetitive P2X7 antagonist

Purity: > 90%

 
 
 
 
Asc-444  

BzATP triethylammonium salt 

Potent, prototypic P2X7 agonist. P2 agonist.

Purity: > 98%

 
Specific publication references
 
 
 
Asc-240  

Caffeine 

PDE inhibitor. Adenosine antagonist

Purity: > 99%

 
 
 
 
Asc-453  

CGS 21680 

Potent, selective A2A agonist

Purity: > 98%

 
 
 
 
Asc-434  

2-Chloro-N6-cyclopentyladenosine (CCPA) 

Highly potent, selective A1 agonist

Purity: > 98%

 
 
 
 
Asc-037  

2-Chloroadenosine (CADO) 

Adenosine agonist

Purity: > 98%

 
Specific publication references
 
 
 
Asc-442  

8-(3-Chlorostyryl)caffeine 

Selective A2A receptor antagonist. MAO-B inhibitor.

Purity: > 98%

 
 
 
 
Asc-387  

(±)-Clopidogrel 

Potent, selective P2Y12 antagonist

Purity: > 99%

 
 
 
 
Asc-472  

N6-Cyclohexyladenosine 

Selective A1 receptor agonist

Purity: > 98%

 
 
 
 
Asc-398  

N6-Cyclopentyladenosine (CPA) 

Potent, selective A1 agonist

Purity: > 99%

 
Specific publication references
 
 
 
Asc-396  

DPCPX 

Potent A1 antagonist

Purity: > 99%

 
Specific publication references
 
 
 
Asc-395  

GW791343 

P2X7 allosteric modulator

Purity: > 99%

 
 
 
 
Asc-458  

HENECA 

Selective A2A receptor agonist

Purity: > 99%

 
 
 
 
Asc-438  

IB-MECA 

Highly potent and selective A3 agonist

Purity: > 97%

 
 
 
 
Asc-421  

KN-62 

CaM kinase II inhibitor. P2X7 antagonist.

Purity: > 98%

Images
 
 
 
 
Asc-397  

MRS 1754 

Selective A2B antagonist

Purity: > 98%

 
 
 
 
Asc-414  

MRS 2179 

Potent, selective P2Y1 antagonist

Purity: > 98%

 
 
 
 
Asc-445  

MRS 2211 

Selective competitive P2Y13 antagonist

Purity: > 95%

 
 
 
 
Asc-440  

NECA 

Highly potent adenosine agonist

Purity: > 99%

 
 
 
 

NECA Fluorescent ligand (Red) 

Fluorescent non-selective adenosine agonist

Purity: > 97%

Images
 
 
 
 
Asc-454  

NF023 

Competitive P2X1 receptor antagonist

Purity: > 97%

 
 
 
 
Asc-415  

NF 449 

Highly selective, potent P2X1 receptor antagonist

Purity: > 95%

 
 
 
 
Asc-403  

β-Nicotinamide adenine dinucleotide (β-NAD) 

Coenzyme and enzyme substrate. P2Y11 agonist.

Purity: > 96%

 
 
 
 
Asc-009  

PPADS 

P2 purinergic receptor antagonist.

 
Specific publication references
 
 
 
Asc-439  

SCH-58261 

Potent, highly selective A2A antagonist

Purity: > 99%

 
 
 
 
Asc-422  

Suramin hexasodium salt 

Non-selective P2 purinergic antagonist

Purity: > 99%

 
Specific publication references
 
 
 

Ticlopidine Hydrochloride 

Selective P2Y12 receptor antagonist

Purity: > 98%

 
 
 
 
Asc-384  

UDP-glucose 

Highly potent P2Y14 agonist

Purity: > 98%

 
 
 
 
Asc-383  

UDP sodium salt (Uridine 5'-diphosphate) 

P2Y6 agonist. P2Y14 ligand.

Purity: > 98%

 
 
 
 
Asc-218  

ZM 241385 

Potent, selective A2A antagonist

Purity: > 99%