Enzyme-Linked Receptors

Code

Name

Details

 Image Abreview Publication 

  

AAL 993 

Potent, selective and cell-permeable VEGFR inhibitor

Purity: > 98%

 
 
 
 
  

(+)-Abscisic acid 

Phytohormone; produced by a variety of cells in humans and animals

Purity: > 99%

 
 
 
 
  

Afatinib (BIBW 2992) 

Potent, irreversible Her2/ErbB 2 and EGFR kinase inhibitor

Purity: > 99%

 
 
 
 
  

AG-370 

Selective PDGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

AG-494 

Potent, selective EGF receptor tyrosine kinase

Purity: > 99%

 
 
 
 
  

AG-1024 

Selective IGF-1 receptor inhibitor. Potent antiproliferative agent.

Purity: > 99%

 
 
 
 
  

AG 1296 

Potent specific PDGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

AG 1478 

Selective EGF receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

AG-879 

Selective TrkA receptor inhibitor

Purity: > 99%

 
 
 
 
  

AMD3100 octahydrochloride 

Highly selective CXCR4 antagonist

Purity: > 99%

 
 
 
 
  

BIBW2992 (Afatinib) 

Potent, irreversible ATP-competitive ErbB inhibitor. Antitumor.

Purity: > 99%

 
 
 
 
  

BMS-599626 (AC480) 

Selective HER1 and HER2 inhibitor

Purity: > 99%

 
 
 
 
  

BX 513 hydrochloride 

Potent and selective CCR1 antagonist

Purity: > 99%

 
 
 
 
  

Canertinib (CI-1033) 

Potent irreversible EGFR and HER2/ErbB2 tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

Celastrol from Celastrus scandens 

Anti-inflammatory and anti-proliferative agent

Purity: > 99%

 
 
 
 
  

Chromium picolinate 

Insulin potentiator

Purity: > 98%

 
 
 
 
  

CP-724714 

Potent, selective HER2/ErbB2 tyrosine kinase inhibitor

Purity: > 95%

 
 
 
 
  

Cryptotanshinone 

STAT3 inhibitor with diverse biological activities

Purity: > 99%

Images
 
 
 
 
  

Diacerein 

Inhibitor of interleukin-1B (IL-1B) production

Purity: > 96%

 
 
 
 
  

7,8-Dihydroxyflavone (7,8-DHF) 

Selective TrkB receptor agonist. Flavonoid.

Purity: > 99%

 
 
 
 
  

DMPQ dihydrochloride 

Potent and selective PDGFRβ inhibitor

Purity: > 99%

 
 
 
 
  

DMXAA (ASA404) 

Vascular disrupting agent. VEGFR inhibitor.

Purity: > 99%

 
 
 
 
  

Erbstatin Analog 

EGFR tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

Gambogic amide 

Potent, selective high affinity nerve growth factor (TrKa) receptor agonist

Purity: > 98%

 
 
 
 
  

Genistein 

Protein tyrosine kinase inhibitor. Anticancer agent.

Purity: > 99%

 
Specific publication references
 
 
 
  

Glipizide 

Sulfonylurea receptor and ATP-sensitive K+ channel blocker

Purity: > 98%

 
 
 
 
  

Glucagon (19-29) (human) 

C-terminal fragment of Glucagon. Potent Ca2+/Mg2+-ATPase inhibitor.

Purity: > 95%

 
 
 
 
  

Gly-Arg-Gly-Asp-Ser 

Synthetic integrin antagonist

Purity: > 98%

 
 
 
 
  

GW 2580 

Selective cFMS RTK inhibitor. Cell-permeable.

Purity: > 99%

 
 
 
 
  

HNMPA-(AM)3 

Insulin receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

ISCK03 

Cell permeable, selective SCF/c-Kit inhibitor

Purity: > 99%

 
 
 
 
  

Ki20227 

Highly selective c-Fms tyrosine kinase inhibitor

Purity: > 95%

 
 
 
 
  

Lestaurtinib 

Potent JAK2, FLT3 and TrkA receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

Leukadherin-1 

Integrin CD11b/CD19 agonist

Purity: > 97%

 
 
 
 
  

(±)-Lisofylline 

Anti-inflammatory agent.

Purity: > 98%

 
 
 
 
  

Luteolin 

Antioxidant, anti-inflammatory, anticancer flavonoid

Purity: > 99%

 
 
 
 
  

LY 364947 

Potent, selective ATP-competitive TGFβ receptor kinase I inhibitor

Purity: > 98%

 
 
 
 
  

Hydroxy-2-naphthalenylmethylphosphonic acid (HNMPA) 

Insulin receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

Nateglinide 

Insulin secretagog agent. K+ channel blocker

 
 
 
 
  

P1 

EGF receptor binding inhibitor

Purity: > 95%

 
 
 
 
  

PD 174265 

Potent, selective, reversible EGFR tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

Pentoxifylline 

Phosphodiesterase inhibitor. Cytokine inhibitor.

Purity: > 99%

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Quizartinib 

Potent, selective Flt3 inhibitor

Purity: > 99%

 
 
 
 
  

RG-14620 

EGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

Royal jelly acid (10-Hydroxy-2-decenoic acid) 

VEGF inhibitor

Purity: > 98%

 
 
 
 
  

SB431542 

ALK inhibitor

Purity: > 99%

 
Specific publication references
 
 
 
  

SU 11274 

Potent, selective cell-permeable Met inhibitor

Purity: > 98%

 
 
 
 
  

SU 6668 

Potent PDGFR inhibitor

Purity: > 98%

 
 
 
 
  

SU 1498 

Selective VEGFR2 inhibitor

Purity: > 98%

 
 
 
 
  

SU4312 

Potent, selective VEGFR and PDGFR receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

SU-5402 

Potent FGFR and VEGFR inhibitor

Purity: > 95%

 
 
 
 
  

SU 5416 (Semaxanib) 

Potent and selective VEGFR inhibitor

Purity: > 99%

 
 
 
 
  

TAK 165 

Potent HER2 tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
  

Tie2 kinase inhibitor 

Potent, reversible and selective ATP-binding site-targeting Tie2 kinase inhibitor. Cell-permeable.

Purity: > 99%

 
 
 
 
  

Tyrphostin 25 (RG-50875) 

Competitive EGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

Tyrphostin 47 

EGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

Tyrphostin 51 

EGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

Tyrphostin 9 

Selective PDGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
  

XL-880 (Foretinib) 

Potent ATP-competitive HGFR and VEGFR2 inhibitor

Purity: > 98%