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Enzyme-Linked Receptors

Code

Name

Details

 Image Abreview Publication 

Lapatinib ditosylate 

Potent PTK inhibitor

Purity: > 99%

 
 
 
 
Asc-860  

(+)-Abscisic acid 

Phytohormone; produced by a variety of cells in humans and animals

Purity: > 99%

 
 
 
 

AG-370 

Selective PDGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

AG-494 

Potent, selective EGF receptor tyrosine kinase

Purity: > 99%

 
 
 
 
Asc-1170  

AG 1296 

Potent specific PDGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

AG 1478 

Selective EGF receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 
Asc-1059  

AG-879 

Selective TrkA receptor inhibitor

Purity: > 99%

 
 
 
 
Asc-718  

AMD3100 octahydrochloride 

Highly selective CXCR4 antagonist

Purity: > 99%

 
 
 
 

BIBW2992 (Afatinib) 

Potent, irreversible ATP-competitive ErbB inhibitor. Antitumor.

Purity: > 99%

 
 
 
 

BMS-599626 (AC480) 

Selective HER1 and HER2 inhibitor

Purity: > 99%

 
 
 
 
Asc-811  

BX 513 hydrochloride 

Potent and selective CCR1 antagonist

Purity: > 99%

 
 
 
 

Canertinib (CI-1033) 

Potent irreversible EGFR and HER2/ErbB2 tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 
Asc-655  

Celastrol from Celastrus scandens 

Anti-inflammatory and anti-proliferative agent

Purity: > 99%

 
 
 
 
Asc-666  

Cryptotanshinone 

STAT3 inhibitor with diverse biological activities

Purity: > 99%

Images
 
 
 
 
Asc-996  

7,8-Dihydroxyflavone (7,8-DHF) 

Selective TrkB receptor agonist. Flavonoid.

Purity: > 99%

 
 
 
 
Asc-1269  

DMPQ dihydrochloride 

Potent and selective PDGFRβ inhibitor

Purity: > 99%

 
 
 
 

Erbstatin Analog 

EGFR tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 

Gambogic amide 

Potent, selective high affinity nerve growth factor (TrKa) receptor agonist

Purity: > 98%

 
 
 
 
Asc-112  

Genistein 

Protein tyrosine kinase inhibitor. Anticancer agent.

Purity: > 99%

 
Specific publication references
 
 
 
Asc-1092  

Gly-Arg-Gly-Asp-Ser 

Synthetic integrin antagonist

Purity: > 98%

 
 
 
 

Lestaurtinib 

Potent JAK2, FLT3 and TrkA receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 

Leukadherin-1 

Integrin CD11b/CD19 agonist

Purity: > 97%

 
 
 
 

(±)-Lisofylline 

Anti-inflammatory agent.

Purity: > 98%

 
 
 
 
Asc-662  

Luteolin 

Antioxidant, anti-inflammatory, anti-cancer flavonoid

Purity: > 99%

 
 
 
 
Asc-725  

Pentoxifylline 

Phosphodiesterase inhibitor. Cytokine inhibitor.

Purity: > 99%

Images
 
 
 
 

RG-14620 

EGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

SU 6668 

Potent PDGFR inhibitor

Purity: > 98%

 
 
 
 

SU4312 

Potent, selective VEGFR and PDGFR receptor tyrosine kinase inhibitor

Purity: > 98%

 
 
 
 

Tyrphostin 25 (RG-50875) 

Competitive EGF receptor tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

Tyrphostin 47 

EGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

Tyrphostin 51 

EGFR tyrosine kinase inhibitor

Purity: > 99%

 
 
 
 

Tyrphostin 9 

Selective PDGFR tyrosine kinase inhibitor

Purity: > 99%