We have 28 products in: Biochemicals >> Pharmacology >> Receptors & Transporters >> Histamine >> H1

Histamine H1 receptors

Code

Name

Details

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Asenapine maleate 

Multiple receptor antagonist. Antipsychotic agent.

Purity: > 99%

 
 
 
 

Astemizole 

Potent, selective histamine H1 receptor antagonist and potent hERG K+ channel blocker

Purity: > 99%

 
 
 
 

Azatadine maleate 

Potent, competitive H1 receptor antagonist. Various pharmacological effects.

Purity: > 98%

 
 
 
 

Azelastine hydrochloride 

Potent and selective H1 receptor antagonist. Potent hERG K+ channel blocker.

 
 
 
 

Betahistine dihydrochloride 

Competitive partial H1 receptor agonist and H3 receptor antagonist

Purity: > 99%

 
 
 
 

Cetirizine dihydrochloride 

Selective histamine H1 receptor antagonist

Purity: > 99%

 
 
 
 

(±)-Chlorpheniramine maleate 

Potent H1 antagonist and SNRI

Purity: > 99%

 
 
 
 

Chlorprothixene 

Potent, non-selective dopamine, 5-HT and H1 receptor antagonist

Purity: > 97%

 
 
 
 

Clemastine Fumarate 

Potent and selective H1 receptor antagonist. Potent HERG K+ channel inhibitor.

Purity: > 99%

 
 
 
 

Clemizole 

Selective H1 receptor antagonist. Antiviral agent.

Purity: > 97%

 
 
 
 

Cyclizine dihydrochloride 

H1 receptor antagonist

Purity: > 99%

 
 
 
 

Cyproheptadine hydrochloride 

Potent H1 and 5-HT2B antagonist. Non-selective receptor antagonist.

Purity: > 99%

 
 
 
 

Desloratadine 

Highly potent, selective H1 receptor antagonist

Purity: > 97%

 
 
 
 

Diphenhydramine hydrochloride 

Potent H1 antagonist

Purity: > 99%

 
 
 
 

Doxepin hydrochloride 

Potent monoamine receptor antagonist and reuptake inhibitor

Purity: > 98%

 
 
 
 

Fexofenadine hydrochloride 

Selective H1 receptor antagonist

Purity: > 99%

 
 
 
 

Histamine dihydrochloride 

Endogenous histamine receptor agonist

 
 
 
 

Hydroxyzine dihydrochloride 

H1 receptor antagonist

Purity: > 98%

 
 
 
 

Levocetirizine dihydrochloride 

Potent and selective H1 receptor antagonist

Purity: > 98%

 
 
 
 

Mepyramine Fluorescent ligand (Red) 

Fluorescent H1 antagonist

Purity: > 97%

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Mepyramine maleate 

Selective H1 inverse agonist

Purity: > 99%

 
 
 
 

Mianserin hydrochloride 

Multiple receptor antagonist. Activity at 5-HT2, H1 and α2 receptors.

Purity: > 99%

 
 
 
 

Mizolastine 

Potent H1 receptor antagonist

Purity: > 99%

 
 
 
 

Olanzapine 

Non-selective 5-HT, dopamine, histamine and muscarinic antagonist

Purity: > 99%

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Orphenadrine hydrochloride 

Nonselective mACh receptor antagonist. H1 and uncompetitive PCP binding site NMDA receptor antagonist. Voltage gated Na+ channel blocker.

Purity: > 96%

 
 
 
 

Terfenadine 

K+ channel blocker. H1 antagonist.

Purity: > 98%

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Tolazoline hydrochloride 

Non-selective, competitive α-adrenoceptor antagonist. Histamine H1 receptor agonist.

Purity: > 99%

 
 
 
 

Tripelennamine Hydrochloride 

H1 receptor antagonist