Selective, competitive P2Y13 antagonist (pA2 = 6.3). Displays >20-fold selectivity over P2Y1 and P2Y12 (IC50 > 10 μM for inhibition of human P2Y1 and human P2Y12 receptor-mediated phospholipase C responses).
2-[(2-Chloro-5-nitrophenyl)azo]-5-hydroxy-6-methyl-3-[(phosphonooxy)methyl]-4-pyridinecarboxaldehyde sodium salt
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months.
Soluble in water to 70 mM
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.