Biological descriptionβ1 Adrenoceptor antagonist. Ki values are 1.14 and 48.7 μM for receptor subtypes β1 and β2, respectively. Antihypertensive. Limited ability to cross the blood-brain barrier.
Storage instructionsStore at Room Temperature. The product can be stored for up to 12 months.
Solubility overviewSoluble in water to 25 mM
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Golf S et al. Relative selectivity of different beta-adrenoceptor antagonists for human heart beta 1- and beta 2-receptor subtypes assayed by a radioligand binding technique. Scand J Clin Lab Invest47:719-23 (1987).
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