Key features and details
- Highly selective, potent κ-opioid agonist
- CAS Number: 112282-24-3
- Purity: > 99%
- Soluble in water to 5 mM and in DMSO to 25 mM (with warming)
- Form / State: Solid
- Source: Synthetic
Product nameBRL 52537 hydrochloride, kappa-opioid agonist
DescriptionHighly selective, potent κ-opioid agonist
Highly selective and potent κ-opioid agonist (Ki = 0.24 nM). 25 times more potent than morphine. Neuroprotective effects seen in vivo.
Chemical name2-(3,4-Dichlorophenyl)-1-[2-(1-pyrrolidinylmethyl)-1-piperidinyl]ethanone hydrochloride
Storage instructionsStore at Room Temperature. The product can be stored for up to 12 months.
Solubility overviewSoluble in water to 5 mM and in DMSO to 25 mM (with warming)
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
ab120669 has not yet been referenced specifically in any publications.