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MW 445.4 Da, Purity >98%. Cell-permeable, competitive, selective, potent p300/CBP histone acetyltransferase inhibitor (Ki = 400 nM). Blocks dynamic acetylation. Anticancer agent. Active in vitro and in vivo.
Alternative names=E1A binding protein p300, E1A-associated protein p300, EP300: E1A binding protein p300, EP300_HUMAN, Histone acetyltransferase p300, KAT3B, RSTS2, p300 HAT
- CAS number
328968-36-1
- Purity
> 98%
- Form
Solid
- Molecular weight
445.4 Da
- Molecular formula
C24H19N3O6
- PubChem identifier
2871948
- Nature
Synthetic
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MW 445.4 Da, Purity >98%. Cell-permeable, competitive, selective, potent p300/CBP histone acetyltransferase inhibitor (Ki = 400 nM). Blocks dynamic acetylation. Anticancer agent. Active in vitro and in vivo.
Alternative names=E1A binding protein p300, E1A-associated protein p300, EP300: E1A binding protein p300, EP300_HUMAN, Histone acetyltransferase p300, KAT3B, RSTS2, p300 HAT
Key facts
- CAS number
328968-36-1
- Purity
> 98%
- Form
Solid
- Molecular weight
445.4 Da
- Molecular formula
C24H19N3O6
- PubChem identifier
2871948
- Nature
Synthetic
- Biochemical name
4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
- Biological description
Cell-permeable, competitive, selective, potent p300/CBP histone acetyltransferase inhibitor (Ki = 400 nM). Blocks dynamic acetylation. Anticancer agent. Active in vitro and in vivo.
- Canonical SMILES
CC1=CC(=C(C=C1C)[N+](=O)[O-])C2=CC=C(O2)C=C3C(=NN(C3=O)C4=CC=C(C=C4)C(=O)O)C
- InChI
InChI=1S/C24H19N3O6/c1-13-10-20(21(27(31)32)11-14(13)2)22-9-8-18(33-22)12-19-15(3)25-26(23(19)28)17-6-4-16(5-7-17)24(29)30/h4-12H,1-3H3,(H,29,30)
- InChIKey
HEKJYZZSCQBJGB-UHFFFAOYSA-N
- IUPAC name
4-[4-[[5-(4,5-dimethyl-2-nitrophenyl)furan-2-yl]methylidene]-3-methyl-5-oxopyrazol-1-yl]benzoic acid
Storage
- Shipped at conditions
Ambient - Can Ship with Ice
- Appropriate long-term storage conditions
-20°C
- Storage information
Store under desiccating conditions, The product can be stored for up to 12 months
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