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MW 482.5 Da, Purity >=98%. IITZ-01 (ab287028) is a potent lysosomotropic autophagy inhibitor; displays >10-fold potent autophagy inhibition than Chloroquine; enhances autophagosome accumulation but inhibits autophagosomal degradation by impairing lysosomal function, finally resulting in the inhibition of autophagy. Displays potent anticancer activity.

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Key facts

CAS number
1807988-47-1
Purity
>= 98%
Form
Solid
Molecular weight
482.5 Da
Molecular formula
C26H23FN8O
PubChem identifier
134817273
Nature
Synthetic

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MW 482.5 Da, Purity >=98%. IITZ-01 (ab287028) is a potent lysosomotropic autophagy inhibitor; displays >10-fold potent autophagy inhibition than Chloroquine; enhances autophagosome accumulation but inhibits autophagosomal degradation by impairing lysosomal function, finally resulting in the inhibition of autophagy. Displays potent anticancer activity.

Key facts

Purity
>= 98%
PubChem identifier
134817273
Solubility

Soluble in DMSO to >100 mM.

Biochemical name
CID 134817273
Biological description

IITZ-01 (ab287028) is a potent lysosomotropic autophagy inhibitor; displays >10-fold potent autophagy inhibition than Chloroquine; enhances autophagosome accumulation but inhibits autophagosomal degradation by impairing lysosomal function, finally resulting in the inhibition of autophagy. Displays potent anticancer activity.

Canonical SMILES
C1COCCN1C2=NC(=NC(=N2)NC3=CC=C(C=C3)F)NC4=CC=C(C=C4)C5=NC6=CC=CC=C6N5
InChI
InChI=1S/C26H23FN8O/c27-18-7-11-20(12-8-18)29-25-32-24(33-26(34-25)35-13-15-36-16-14-35)28-19-9-5-17(6-10-19)23-30-21-3-1-2-4-22(21)31-23/h1-12H,13-16H2,(H,30,31)(H2,28,29,32,33,34)
InChIKey
XGEDDGLPNSLBFE-UHFFFAOYSA-N
IUPAC name
4-N-[4-(1H-benzimidazol-2-yl)phenyl]-2-N-(4-fluorophenyl)-6-morpholin-4-yl-1,3,5-triazine-2,4-diamine

Storage

Shipped at conditions
Blue Ice
Appropriate long-term storage conditions
-20°C

Notes

This product is manufactured by BioVision, an Abcam company and was previously called B2378 IITZ-01. B2378-5 is the same size as the 5 mg size of ab287028.

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