IPA 3, Group I, p21-activated kinase (PAK) inhibitor
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(1 Publication)
MW 350.5 Da, Purity >97%. Group I, p21-activated kinase (PAK) inhibitor (IC50 = 2.5 μM). Non-ATP competitive, allosteric inhibition in vivo. Selectivity over >200 other kinases.
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1 25 dihydroxyvitamin D3 receptor, 25-dihydroxyvitamin D3 receptor, CBX, CBX1_HUMAN, Chromobox 1, Chromobox homolog 1 (HP1 beta homolog Drosophila ), Chromobox protein homolog 1, Drosophila HP1 beta, ERR a, ERR-alpha, ERR1 protein, ERR1_HUMAN, ESRL 1, ESRR A, Estrogen receptor related 1, Estrogen receptor-like 1, Estrogen-related receptor alpha, Estrra, FH, FUMH_HUMAN, Fumarase, Fumarate hydratase, Fumarate hydratase mitochondrial, HLRCC, HP1 beta, HP1 beta homolog, HP1 beta homolog Drosophila, HP1, Drosophila. homolog of, beta, HP1Hs beta, Heterochromatin protein 1 beta, Heterochromatin protein 1 homolog beta, Heterochromatin protein p25, Human heterochromatin protein p25 mRNA complete cds, LRCC, M31, MCL, MCUL 1, MGC2124, MGC60244, MOD 1, MS709, Member 1, Modifier 1 protein, Multiple hereditary cutaneous leiomyomata, NR1I1, NR3B1, Nuclear receptor subfamily 1 group I member 1, Nuclear receptor subfamily 3 group B member 1, PPP1R163, Protein phosphatase 1, regulatory subunit 163, RGP 4, RGS4_HUMAN, Regulator of G protein signalling 4, Regulator of G-protein signaling 4, SCZD 9, Schizophrenia disorder 9, Steroid hormone receptor ERR1, VDR_HUMAN, Vitamin D (1,25- dihydroxyvitamin D3) receptor, Vitamin D hormone receptor, Vitamin D nuclear receptor variant 1, Vitamin D receptor, Vitamin D3 receptor, chromobox homolog 1, estrogen receptor related receptor alpha, hERR1, heterochromatin protein p25 beta, p25beta
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Chemical Structure - IPA 3, Group I, p21-activated kinase (PAK) inhibitor (AB141014)
2D chemical structure image of ab141014, IPA 3, Group I, p21-activated kinase (PAK) inhibitor
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Publications (1)
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World journal of gastroenterology 21:9945-56 PubMed26379399
2015
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