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MW 511.6 Da, Purity >95%. MMP-9 inhibitor. Role in tumor cell migration, invasion and angiogenesis. Achieve your results faster with highly validated, pure and trusted compounds.

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Publications

Key facts

CAS number
1177749-58-4
Purity
> 95%
Molecular weight
511.6 Da
Molecular formula
C27H33N3O5S
PubChem identifier
21310926
Nature
Synthetic

Alternative names

Recommended products

MW 511.6 Da, Purity >95%. MMP-9 inhibitor. Role in tumor cell migration, invasion and angiogenesis. Achieve your results faster with highly validated, pure and trusted compounds.

Key facts

Purity
> 95%
PubChem identifier
21310926
Solubility

Soluble in DMSO to 10 mM.

Biochemical name
MMP-9 Inhibitor I
Biological description

MMP-9 inhibitor. Role in tumor cell migration, invasion and angiogenesis

Canonical SMILES
CCN(CC)CC1=CC(=C(C(=C1)C)N(CC2=CC=CC=C2)S(=O)(=O)C3=CC=C(C=C3)OC)C(=O)NO
InChI
InChI=1S/C27H33N3O5S/c1-5-29(6-2)18-22-16-20(3)26(25(17-22)27(31)28-32)30(19-21-10-8-7-9-11-21)36(33,34)24-14-12-23(35-4)13-15-24/h7-17,32H,5-6,18-19H2,1-4H3,(H,28,31)
InChIKey
WRNMBFWQBKEBIX-UHFFFAOYSA-N
IUPAC name
2-[benzyl-(4-methoxyphenyl)sulfonylamino]-5-(diethylaminomethyl)-N-hydroxy-3-methylbenzamide

Storage

Shipped at conditions
Ambient - Can Ship with Ice
Appropriate short-term storage conditions
-20°C
Appropriate long-term storage conditions
-20°C
Storage information
Store under desiccating conditions, The product can be stored for up to 12 months

Notes

This product is manufactured by BioVision, an Abcam company and was previously called 1981 MMP-9 Inhibitor. 1981-500 is the same size as the 500 μg size of ab142180.

Supplementary info

This supplementary information is collated from multiple sources and compiled automatically.
Activity summary

The proteins MMP1 MMP9 and MMP13 belong to the matrix metalloproteinase (MMP) family and function mainly as enzymes that degrade various components of the extracellular matrix. MMP1 also known as collagenase-1 has a mass of approximately 54 kDa and primarily targets interstitial collagen. MMP9 known as gelatinase B is about 92 kDa and digests denatured collagen (gelatin) and elastin. MMP13 or collagenase-3 is around 60 kDa and degrades type II collagen among other substrates. These MMPs express in various tissues including skin cartilage and the immune system playing roles in tissue remodeling and repair.

Biological function summary

These MMPs regulate extracellular matrix composition and influence cellular behaviors like migration and invasion. MMP1 MMP9 and MMP13 participate in normal developmental processes and the breakdown of extracellular matrix in pathological conditions. They form complexes with tissue inhibitors of metalloproteinases (TIMPs) that modulate their activities ensuring balanced matrix turnover. Their expression requires precise control because unregulated activity can lead to tissue damage.

Pathways

MMP1 MMP9 and MMP13 integrate into complex networks like the collagen degradation and inflammation pathways. MMP9 is an important actor in the inflammatory response often upregulated by cytokines and serving a role in leukocyte migration facilitated by its interaction with integrins. The Wnt signaling pathway connects to MMP13 highlighting its involvement in cartilage metabolism and bone remodeling. These proteins interact with others in these pathways like interleukins and integrins to coordinate a broad range of physiological effects.

Associated diseases and disorders

MMP dysregulation associates with conditions like arthritis and cancer. In arthritis MMP13 excessively degrades cartilage collagen contributing to joint destruction while interactions with cytokines amplify inflammation. In cancer MMP9 assists tumor invasion and metastasis through matrix degradation and works in conjunction with VEGF to promote angiogenesis. MMP9 inhibitors have been investigated for therapeutic use in cancer treatment due to these contributions. Understanding these mechanisms highlights the importance of MMP regulation and inhibition in disease contexts.

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