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Epsin-1

Domain

The NPF repeat domain is involved in EPS15 binding.

The DPW repeat domain is involved in AP2A2 and clathrin binding.

The [DE]-X(1,2)-F-X-X-[FL]-X-X-X-R motif mediates interaction with the AP-2 complex subunit AP2B1.

Function

Binds to membranes enriched in phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2). Modifies membrane curvature and facilitates the formation of clathrin-coated invaginations (By similarity). Regulates receptor-mediated endocytosis (PubMed:10393179, PubMed:10557078).

Post-translational modifications

Phosphorylated on serine and/or threonine residues in mitotic cells. Phosphorylation reduces interaction with REPS2, AP-2 and the membrane fraction. Depolarization of synaptosomes results in dephosphorylation.

Ubiquitinated.

Sequence Similarities

Belongs to the epsin family.

Cellular localization

Alternative names

Epsin-1, EH domain-binding mitotic phosphoprotein, EPS-15-interacting protein 1, EPN1

swissprot:Q9Y6I3 entrezGene:29924 omim:607262