Key features and details
- Selective galanin GAL2 receptor antagonist
- CAS Number: 908844-75-7
- Soluble in water
- Form / State: Solid
- Source: Synthetic
Product nameM871, Galanin GAL2 receptor antagonist
DescriptionSelective galanin GAL2 receptor antagonist
Selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively). Blocks pronociceptive effects of GAL2 agonists including AR-M1896. Active in vivo.
SequenceWTLNSAGYLLGPEHPPPALALA (Modifications: C-terminal amide)
Storage instructionsStore at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months.
Solubility overviewSoluble in water
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
ab141159 has been referenced in 1 publication.
- Lin CY et al. Spexin Enhances Bowel Movement through Activating L-type Voltage-dependent Calcium Channel via Galanin Receptor 2 in Mice. Sci Rep 5:12095 (2015). PubMed: 26160593