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Home Agonists, activators, antagonists and inhibitors

Enzyme modulators

Product
  • ATPase & GTPase
  • Caspase
  • Cyclases
  • Kinase
  • Phosphatases
  • Proteases

Enzyme activators and inhibitors are essential in the study of intracellular mechanisms. The presence of these modulators may lead to an alteration in biological activity, with the effect being dependent on the use of an activator or inhibitor. Popular enzymes include PI3K/Akt, MAPK and JAK-STAT, many of which form cell signaling pathways. Join researchers worldwide and find enzyme modulators for your research.

Browse all related products

Features

MAPK pathway​​

Download our guide to the MAPK pathway highlighting the proteins responsible for cellular communication.

Advantages of small molecule inhibitors

Our guide written by Professor Stephen Taylor highlights the opportunities for you of using inhibitors.

Guidelines for small-molecule inhibitors

Choose the right inhibitor for your experiment by reading our guide written by Professor Stephen Taylor.



  • All
  • Articles
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  • Protocols

Protocols and troubleshooting tips, to help get the best from our antibodies

637497563610000000

Protocol

Western blot FAQ

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Protocol

Abreview

Abreviews®, our peer review program

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Article

Western blot troubleshooting tips

637431061250000000

Protocol

Advantages of small-molecule inhibitors

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Actin filament polymerization

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Article

Dorsomorphin (Compound C), AMP-kinase inhibitor (ab120843)

636899934910000000

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Z-VAD(OMe)-FMK, Cell permeable, irreversible pan-caspase inhibitor (ab120487)

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Z-VAD(OH)-FMK, Irreversible general caspase inhibitor (ab120382)

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Forskolin, Adenylyl cyclase activator (ab120058)

636899932530000000

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Dyngo® 4a, Novel, highly dynamin inhibitor (ab120689)

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SP600125, JNK inhibitor (ab120065)

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Mertansine (DM1 Compound), microtubule-targeted cytotoxic agent (ab146096)

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8-(4-Chlorophenylthio)adenosine 3',5'-cyclic monophosphate (8-CPT-cAMP), Cell permeable cAMP analog. (ab120424)

636899916690000000

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NKH 477 (Colforsin daropate), an adenylyl cyclase activator (ab120190)

636899915730000000

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SU 5416 (Semaxanib), VEGFR-2 inhibitor (ab145056)

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AICAR (Acadesine/AICA riboside), AMPK activator (ab120358)

636899914610000000

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MG-132, proteasome inhibitor (ab141003)

636899914100000000

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Okadaic acid, PP1 and PP2A inhibitor (ab120375)

636899913150000000

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Dynasore, dynamin inhibitor (ab120192)

636899912570000000

Product

A 769662, AMP-activated protein kinase activator (ab120335)

636899911850000000

Product

Bafilomycin A1, (V)-ATPase inhibitor (ab120497)

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Product

Y-27632 dihydrochloride (ab120129)

636899879550000000

Product

Thapsigargin (ab120286)

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Product

Phorbol 12-myristate 13-acetate (PMA) (ab120297)

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Product

Staurosporine (ab120056)

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Guidelines for small-molecule inhibitors.

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Article

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