Overview

  • Product name

    Zamifenacin fumarate, M3 receptor antagonist
  • Description

    Selective M3 receptor antagonist
  • Biological description

    Selective M3 receptor antagonist (pKi values are 8.52 (M3), 7.93 (M2), 7.90 (M1) and 7.78 (M4) respectively). Inhibits gastrointestinal motility in vivo without causing cardiovascular effects.
  • Purity

    > 99%
  • CAS Number

    127308-98-9
  • Chemical structure

    Chemical Structure

Properties

References

This product has been referenced in:

  • Choppin A & Eglen RM Pharmacological characterization of muscarinic receptors in dog isolated ciliary and urinary bladder smooth muscle. Br J Pharmacol 132:835-42 (2001). Read more (PubMed: 11181424) »
  • Choppin A  et al. Characterization of the muscarinic receptor in isolated uterus of sham operated and ovariectomized rats. Br J Pharmacol 127:1551-8 (1999). Read more (PubMed: 10455309) »
  • Watson N  et al. Characterization of the interaction of zamifenacin at muscarinic receptors in vitro. Eur J Pharmacol 285:135-42 (1995). Read more (PubMed: 8566131) »

Customer reviews and Q&As

There are currently no Customer reviews or Questions for ab141511.
Please use the links above to contact us or submit feedback about this product.

Please note: All products are "FOR RESEARCH USE ONLY. NOT FOR USE IN DIAGNOSTIC PROCEDURES, NOT FOR USE IN HUMANS"
For licensing inquiries, please contact partnerships@abcam.com

Sign up